Showing posts with label Damiana. Show all posts
Showing posts with label Damiana. Show all posts

Tuesday, April 12, 2016

Natural Ways to Reduce Estrogen Dominance

 
#helpYOUgetGAINS 
Twitter: @helpYOUgetGAINS


DIM


In healthy young men, it cuts "bad" estrogens in half by helping the liver neutralize them. DIM doesn't actually reduce estrogens. What is does is help the liver convert them into weaker forms.


Take 200-300 mg as 2-3 divided doses.


Calcium-D-Glucarate


Calcium D-glucarate attaches itself to estrogens in your intestines and passes them out into your toilet bowl. Otherwise, your body's could reabsorb a significant amout of estrogens that your body intends to eliminate. The only possible downside is that it also helps remove excess testosterone and cortisol, but only the overspill that's already destined for elimination. Take 800-600 mg as 2-8 divided doses.

Damiana Extract

University of Mississippi (Oxford) researchers discovered that damiana leaf extract inhibits the aromatase enzyme that converts testosterone into estrogen in the body. Take 50-500 milligrams three times per day between meals.

Chrysin

5, 7-dihydroxyflavone or chrysin is a flavonoid compound found in many plants and in honey. It has been known for years to inhibit the aromatase enzyme and block the conversion of testosterone into estrogen. Recent research from Texas Tech University (Lubbock) finds that it can also directly increase testosterone production. Take 1 gram of chrysin with breakfast, lunch and dinner.

Methoxyisoflavone

Is an anti-estrogen supplement. It lowers estrogen promoting higher testosterone levels. It also has been found to enhance protein synthesis and lower cortisol levels. Take 500-2,000mg per day in three divided doses with meals

Indole-3-carbinol (I3C)

A closely related derivative diindolylmethane (DIM), naturally occurring phytochemicals also reduces the strength of estrogens by converting them to weaker varieties in the liver.

The new entry's (most are natural ingredients that bind to estrogen receptors):

Resveratrol

Known as the ingredient from the French paradox, resveratrol is a SERM type product that has many other health promoting benefits. Resveratrol has been shown in studies to not only block estrogen but and increase LH leading to higher testosterone levels.

Ellagic Acid

This is typically an extract of raspberries and pomegranate. It has been studied to block estrogen.

Daidzein

This is the soy paradox. We typically say don't take soy. Daidzein which is a metabolite of soy that has weak estrogenic activity.

Grape Seed Extract.

Many studies have shown Grape Seed Extract to be a good aromatase inhibitor.

URSOLIC ACID
This poly phenol found in the skin of apples has been shown to increase muscle growth and strength by increasing production of IGF-1 and reducing the amount of testosterone that gets converted to estrogen. It has also been shown to increase fat loss while simultaneously building more muscle. Take 250-l,500mg 30-60 minutes before workouts.



Ipriflavone or 7-hydroxyflavone

Doses equivalent to about 500 mg for humans, easily reachable with lpriflavone supplements. Studies have found that serum testosterone levels increased, estrogen levels decreased, and muscle RNA went up 5%-10% (meaning more muscle protein was being directed) due to aromatase inhibition.





Stinging nettle

Ori Hofmekler (The Warrior Diet) lists this as having anti-aromatase agent. I will have to do further research.

Safflower Seed

Carthamus tinctorius (Compositae) as an anti-estrogenic. Studies have shown that tracheloside significantly decreased the activity of alkaline phosphatase (AP), an estrogen-inducible marker enzyme. As such CLA has also been pro ported to have anti-estrogenic capabilities.

VITEX AGNUS CASTUS

Chaste tree or Vitex agnus castus contains the active compounds known as agnosides that work to reduce estrogen levels and boost luteinizing hormone (LH) levels. In males, this can lead to a dramatic increase in testosterone. Take 200-400 mg of vitex agnus castus or chasteberry extract immediately before bed. Take it in 6-8-week cycles, then lay off for about four weeks before starting the next cycle.

Citrus Bioflavonoids

Hesperetin is created by metabolising hesperidin in the stomach which is found in citrus fruits, especially orange. Naringenin is another citrus bioflavonoid whose metabolites are able to lower aromatase enzyme and estrogen. They do this by attaching to receptor sites.

Bee Propolis

Has been shown to be effective in the fight against xenoestrogens.

Vitamin D

Has been shown to be a natural aromatase inhibitor.

Turmeric

Has promise as an aromatase inhibitor by occupying estrogen receptors. 








Sources:

Damiana + chrysin: stack these two aminos to send nitric oxide levels skyrocketing.  Jim Stoppani.
Flex. 27.9 (Nov. 2009): p132.

"Grow your chest, not your breasts." Men's Fitness July 2002: 66+.

Your T, on E. Murphy, Myatt. Men's Health, Sep2012, Vol. 27 Issue 7, p86-87, 2p

ERADICATE ESTROGEN TO FUEL YOUR GROWTH. Rowley, Brian. Stoppani, Jim. Joe Weider's Muscle & Fitness, Oct2003, Vol. 64 Issue 10, p176

ESTROGEN NATION. Lockwood, Chris. Joe Weider's Muscle & Fitness, Nov2009, Vol. 70 Issue 11, p94-97


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 You have power over your mind - not outside events. Realize this, and you will find strength ~ Marcus Aurelius

Tuesday, June 10, 2014

SD Pharmaceuticals’ ACACETIN 99™ is a novel new anti-aromatase

ACACETIN 99 - HIGH-QUALITY ACACETIN

SD Pharmaceuticals’ ACACETIN 99™ is a pure form of Acacetin derived from the Damiana (Turnera diffusa) plant. ACACETIN 99™ was developed based on the findings of recent research that examined the anti-aromatase properties of compounds isolated from the Damiana plant!
Anti-Aromatase Estrogen Blocker

WHAT IS ACACETIN?

Acacetin is a natural flavone that is found in the Damiana (Turnera diffusa) plant. Acacetin has been studied for a variety of reasons and some research suggests it may have anti-aromatase and anti-estrogen properties!

HOW DOES ACACETIN WORK?

Research suggests that Acacetin has anti-aromatase properties. Aromatase is the enzyme responsible for converting testosterone to estrogen. Inhibition of the aromatase enzyme helps reduce the amount of testosterone that gets converted to estrogen. Healthy regulation of the aromatase enzyme can help support healthy testosterone and estrogen levels!

STACK WITH TESTOSTERONE BOOSTERS!

Since ACACETIN 99™ is scientifically designed to help reduce aromatase activity it may help reduce the conversion of testosterone to estrogen. That’s why it makes for a great option to stack with testosterone-boosting ingredients!

ACACETIN 99™ - Anti-Estrogen Supplement

Anti-Aromatase Supplement Anti-Estrogen Testosterone Booster

Tuesday, November 6, 2012

Manage Estrogen to Raise Testosterone. SERMs: Anti-Estrogen and Anti-Aromatase Products

Aromatase is an enzyme which converts testosterone to estrogen. Inhibiting aromatase increases testosterone and reduces estrogen, promoting muscle growth and fat loss. Numerous studies have seem to have confirmed this.

In this post I will look at a few of the current means of estrogen management. Often referred to as SERMs or Selective Estrogen Receptor Modulators.

Before with get to the current popular ingredients, let's talk about lifestyle things you can do. These are especially important if you belong to the "big belly club" like me.

  • Lift heavy to build more muscle and burn more glycogen. Less glycogen stores means more body fat burned. 
  • Avoid soy, wheat and flax. Yeah, I know, it's probably bro science but why take a chance. Especially if you are already estrogen prone. 
  • Get 8 hours of sleep. 
  • Avoid alcohol. 
  • Get some. If you don't know what some is.....you already may have lost the fight. 
  • Avoid plastic containers. Water bottles and heating food in plastics. BPA has estrogenic effects. 
  • Eat proteins and don't be afraid of saturated fats. Whole eggs. At least 1 gram per pound of lean body weight. If you weight 200 pounds but you are 30% body fat, don't eat 200 grams of protein. Your lean mass is closer to 140 to 150 pounds lean. About 20 to 30% of your calories should come from fat. 
  • Eat 2 grams of carbs per pound of body weight or less. Learn your body. I'm king endomorph I need to eat less. Most dudes can eat a 2 to 1 ratio of carbs to protein. 
  • If you are a lean dude. No belly and no moobs. Don't worry about estrogen.
  • Eat broccoli and other cruciferous vegetables such as cauliflower and cabbage. They are powerful estradiol blockers.
Now to the individual supplements.





The old standbys:


DIM


In healthy young men, it cuts "bad" estrogens in half by helping the liver neutralize them. DIM doesn't actually reduce estrogens. What is does is help the liver convert them into weaker forms.


Take 200-300 mg as 2-3 divided doses.


Calcium-D-Glucarate


Calcium D-glucarate attaches itself to estrogens in your intestines and passes them out into your toilet bowl. Otherwise, your body's could reabsorb a significant out of estrogens your body intends to eliminate. The only possible downside is that it also helps remove excess testosterone and cortisol, but only the overspill that's already destined for elimination. Take 800-600 mg as 2-8 divided doses.


Damiana Extract


University of Mississippi (Oxford) researchers discovered that damiana leaf extract inhibits the aromatase enzyme that converts testosterone into estrogen in the body. Take 50-500 milligrams three times per day between meals.


Chrysin


5, 7-dihydroxyflavone or chrysin is a flavonoid compound found in many plants and in honey. It has been known for years to inhibit the aromatase enzyme and block the conversion of testosterone into estrogen. Recent research from Texas Tech University (Lubbock) finds that it can also directly increase testosterone production. Take 1 gram of chrysin with breakfast, lunch and dinner.

Methoxyisoflavone

Is an anti-estrogen supplement. It lowers estrogen promoting higher testosterone levels. It also has been found to enhance protein synthesis and lower cortisol levels. Take 500-2,000mg per day in three divided doses with meals

Indole-3-carbinol (I3C)

A closely related derivative diindolylmethane (DIM), naturally occurring phytochemicals also reduces the strength of estrogens by converting them to weaker varieties in the liver.

The new entry's (most are natural ingredients that bind to estrogen receptors):

Resveratrol

Known as the ingredient from the French paradox, resveratrol is a SERM type product that has many other health promoting benefits. Resveratrol has been shown in studies to not only block estrogen but and increase LH leading to higher testosterone levels.

Ellagic Acid

This is typically an extract of raspberries and pomegranate. It has been studied to block estrogen.

Daidzein

This is the soy paradox. We typically say don't take soy. Daidzein which is a metabolite of soy that has weak estrogenic activity.

Grape Seed Extract.

Many studies have shown Grape Seed Extract to be a good aromatase inhibitor.

URSOLIC ACID
This poly phenol found in the skin of apples has been shown to increase muscle growth and strength by increasing production of IGF-1 and reducing the amount of testosterone that gets converted to estrogen. It has also been shown to increase fat loss while simultaneously building more muscle. Take 250-l,500mg 30-60 minutes before workouts.

Ipriflavone or 7-hydroxyflavone

Doses equivalent to about 500 mg for humans, easily reachable with lpriflavone supplements. Studies have found that serum testosterone levels increased, estrogen levels decreased, and muscle RNA went up 5%-10% (meaning more muscle protein was being directed) due to aromatase inhibition.

Stinging nettle

Ori Hofmekler (The Warrior Diet) lists this as having anti-aromatase agent. I will have to do further research.

Safflower Seed

Carthamus tinctorius (Compositae) as an anti-estrogenic. Studies have shown that tracheloside significantly decreased the activity of alkaline phosphatase (AP), an estrogen-inducible marker enzyme. As such CLA has also been pro ported to have anti-estrogenic capabilities.

VITEX AGNUS CASTUS

Chaste tree or Vitex agnus castus contains the active compounds known as agnosides that work to reduce estrogen levels and boost luteinizing hormone (LH) levels. In males, this can lead to a dramatic increase in testosterone. Take 200-400 mg of vitex agnus castus or chasteberry extract immediately before bed. Take it in 6-8-week cycles, then lay off for about four weeks before starting the next cycle.

Citrus Bioflavonoids

Hesperetin is created by metabolising hesperidin in the stomach which is found in citrus fruits, especially orange. Naringenin is another citrus bioflavonoid whose metabolites are able to lower aromatase enzyme and estrogen. They do this by attaching to receptor sites.

Bee Propolis

Has been shown to be effective in the fight against xenoestrogens.

Vitamin D

Has been shown to be a natural aromatase inhibitor.

Turmeric

Has promise as an aromatase inhibitor by occupying estrogen receptors. 





 

Previous Posts:

Cutting Stack: BPI Sports A-HD and Solid

Contest Drawing: Enter to Win BPI Sports A50 and A-HD Stack. Get a headstart on your mass stack.


Sources:

Damiana + chrysin: stack these two aminos to send nitric oxide levels skyrocketing.  Jim Stoppani.
Flex. 27.9 (Nov. 2009): p132.

"Grow your chest, not your breasts." Men's Fitness July 2002: 66+.

Your T, on E. Murphy, Myatt. Men's Health, Sep2012, Vol. 27 Issue 7, p86-87, 2p

ERADICATE ESTROGEN TO FUEL YOUR GROWTH. Rowley, Brian. Stoppani, Jim. Joe Weider's Muscle & Fitness, Oct2003, Vol. 64 Issue 10, p176

ESTROGEN NATION. Lockwood, Chris. Joe Weider's Muscle & Fitness, Nov2009, Vol. 70 Issue 11, p94-97


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Monday, September 3, 2012

7 Steps to Higher Testosterone


High T. Everyman wants it. It means power, energy, virility culminating in the ultimate swagger man. After the age of 30 your testosterone levels begin to drop and continue to drop. Nice thought. If you are under 30 then you don't need the seven steps, just follow the first two.

The normal range is 300-1,200 ng/dL. Typically low testosterone is considered below 280 ng/dL, but most will say that if you drop below 400 you need help.

How do you achieve it? Diet and exercise of course are the platform for your launch. Decreasing fat stores and keeping stress hormones at bay also will help.

There are seven steps you need to complete in order to maximize your testosterone production and use.
Yup, “Ancient Sea Salt” would be a scientifically accurate branding for ordinary table salt.
— Neil deGrasse Tyson (@neiltyson) August 16, 2015

I'm not the most verbose dude so let's jump right in.

1) Eat for Higher T.
    Eat like a freakin man. Whole eggs, beef, nuts. Almonds, brazil nuts and
    cod liver oil. Avocados and olives. Oysters if you can handle it. The
    saturated fat is required. The body uses cholesterol to produce testosterone.
    Sprinkle in a few servings of cruciferous vegetables (broccoli, cabbage, kale
    and collards) keeps your testosterone from becoming estrogen. Grass fed
    beef contains higher levels of CLA which has some value for fat burning
    and anti-aromataze. Drink black tea or real cocoa they lowers cortisol.
    Add wheat germ to your shakes to get teste supporting zinc. Raw honey
    containing atleast 25mg of royal jelly.

2) Lift Heavy and Lift Late
    Heavy compound movements (either heavy 6-8 reps or high reps with
    short rest). Squats and deadlifts should lead the way. Pull-ups, shoulder
    press, bench press, bent-over rows. Why late? Because the stress
    hormone cortisol is higher in the morning and the higher your cortisol
    the lower your testosterone.

3) Increase Luteinizing Hormone (LH). 
Take one of the following. Go five days on/two days off for eight weeks, then take  two weeks off.

    Tribulus terrestris - Take 500-2,000 mg per day in 2-3 divided doses. One dose 30-60 minutes pre-workout.

    D-Aspartic Acid - 3 grams first thing in the morning

    Fenugreek Extract - Take 500-2,000 mg per day.

    Avena sativa -100-250 mg 1-2 times per day, with one dose about 30-60 minutes before your workout.
        
4) Stimulate the Testicles Leydig Cells. 
Go five days on/two days off for eight weeks, then take two weeks off.

     Eurycoma longifolia Jack (Longjax aka Tongkat ali) - 200-300 mg 2 -3 times per day.

     Forskolin (Coleus forskohlii) - Take 20-50 mg 2-3 times daily.

5) Prevent Aromatase (what good is testosterone if it converts into estrogen)
     
Chrysin (also known as 5,7-di-hydroxyflavone) - 1g with breakfast, lunch,  and the last meal of the day
     
Damiana extract - 50-500mg of three times per day in between meals

Diindole or Diindolylmethane (DIM) - 200-300mg in two or three divided doses

6) Free the Testosterone - testosterone can't enter muscle unless it's free from sex-hormone-binding globulin (SHBG)

    Stinging nettle root (urtica dioica) - 100-500 mg of stinging nettle root extract 2-3 times per day on an empty stomach.

    Boron - 10 mg per day was shown to increase free testosterone by almost 30% while also lowering estradiol goes down by forty percent.

    Avena Sativa - see step 3

    Eurycoma longifolia Jack (Longjax aka Tongkat ali) - see step 4
    
7) Increase Your Androgen Receptors - that free testosterone now has to enter muscle tissue.

Carnitine - 1-3 grams of  in the form of L-carnitine, acetyl-L-carnitine or L-carnitine-L-tartrate with breakfast and pre and post workout.

Oh yeah, use alcohol in moderation and have sex frequently. It may be tough to do both since they often go together but do your best.

Remember, this is just advice (like the TMW says), "Do whatever you want to do?"

Bonus information:

Take ZMA - the trio of zinc, magnesium aspartate and vitamin B6 increased testosterone by more than 30% and IGF-1 by 4%.

Blunt cortisol - Higher cortisol means lower testosterone.


Take 5-10 grams of BCAAs in the morning or 800 mg Phosphatidylserine (PS).


Additional information:

How is testosterone made?

From Muscle and Fitness
Stoppani, Jim. "The testosterone diet: finally, a meal plan with one utterly important muscle-building goal: to ramp up your body's levels of testosterone.(NUTRITION). ." Joe Weider's Muscle & Fitness. 67.7 (July 2006): 150(6).

"To understand how diet affects testosterone levels, you first must understand testosterone production and its actions. It all begins in the brain. A hormone called gonadotropin-releasing hormone (GnRH) is released from the hypothalamus (a small section deep within the brain) and travels to the pituitary gland. From here, GnRH stimulates the release of luteinizing hormone, which travels via the blood all the way to the testes, where it activates enzymes that convert cholesterol into testosterone. What you eat can positively or negatively affect any one of these steps.

Your nutritional regimen can also influence testosterone after it's produced. Testosterone travels in the blood to muscle cells and other tissues either as free (or active) testosterone or bound to a carrier protein. Only the free kind can work to increase muscle size by entering the muscle cells. At some tissues, such as fat cells and the brain, fat can be converted into estrogens--yes, the female hormone you don't want in excess in your body, since it can lead to fat gain and inhibit further testosterone production by decreasing brain hormones. Diet can influence the amounts of both active testosterone and estrogens in the blood."
End of Muscle and Fitness excerpt.

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Sources:
Kadey, Matthew."$#'t you can add to shakes: boost testosterone, burn fat or gain energy with a few hassle-free, supercharged additions to your regular protein drink. " Joe Weider's Muscle & Fitness. 71.13 (Dec 2010): 172(5).

Aceto, Chris."Bodybuilding food alternatives: twelve surprising muscle-building foods. " Flex.   23.5 (July 2005): 90(4).

Vittek, J., and B. L. Slomiany. "Testosterone in royal jelly. " Experientia. 40.1 (Jan 1984): 104(3).

Stoppani, Jim. "Aspire to boost test: use the amino acid D-asp to raise testosterone levels. " Flex. 28.8 (Oct 2010): 113(2).

Stoppani, Jim, and Steve Stiefel. "Test drive: dramatically boost your testosterone levels and muscle gains with this six-week training, nutrition and supplement program. " Flex. 23.11 (Jan 2006): 96(9).


 Scheett, Tim. HIGHER TEST SCORES. Joe Weider's Muscle & Fitness (0744-5105) 20071201. Vol.68,Iss.12;p.243-243

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The encyclopedia of supplements. Flex (8750-8915) 1 Feb 2012. p.270(7)

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Breakfast boron capsule boosts testosterone from ergo-log.com

Naghii et al., 2011. Comparative effects of daily and weekly boron supplementation. J Trace Elem Med Bio. 25(1):54-58.